Wednesday, 11th September 13th Australian Peptide Conference 2019
Breakfast
6:30AM - 8:30AM
Wednesday, 11th September
Oak & Vine
GPCRs & Pharmacology
8:30AM - 10:30AM
Wednesday, 11th September
Manhattan Room
Chairs: Ross Bathgate & Anne Conibear
Sponsored by:
- Using cryo-EM to understand peptide GPCR structure function - Patrick Sexton
- Understanding allosteric modulation of GPCRs through structural biology - David Thal
- Crosslinking furan-modified peptides for GPCR target identification on live cells - Laia Miret Casals
- Animal toxins and GPCRs, a promising combination for science and medicine - Nicolas Gilles
- Activation of the relaxin receptor RXFP1 is by a tethered agonist - Paul R. Gooley
- Studying the molecular pharmacology of peptide- and protein-activated receptors - Kevin Pfleger
Morning Tea
10:30AM - 11:00AM
Wednesday, 11th September
Manhattan Foyer
Peptide Chemistry II
11:00AM - 1:00PM
Wednesday, 11th September
Manhattan Room
Chairs: Brad Pentelute & Aline Dantas
Sponsored by:
- Peptide-Based Therapeutics: Paving the Way from the Lab to the Clinic - Margaret Brimble
- A synthetic platform for the generation of anticoagulant sulfoproteins libraries - Emma E Watson
- Design and Synthesis of 13-membered Cyclic Tetrapeptides as Novel Antimicrobials with Enhanced Therapeutic Window - Vijayalekshmi Sarojini
- Biased Inteleukin-1 Receptor Allosteric Modulation with Lactam Peptides for Mitigating Inflammation without Compromising Immuno-Vigilance - William Lubell
- Semi-synthesis of Homogeneous Glycoproteins - Yasuhiro Kajihara
Lunch
1:00PM - 2:00PM
Wednesday, 11th September
Oak & Vine
Free Time
2:00PM - 3:00PM
Wednesday, 11th September
Chemical Biology
3:00PM - 5:00PM
Wednesday, 11th September
Manhattan Room
Chairs: Lara Malins & Laszlo Otvos
- Tools and methods for probing the biology of tryptophan C-mannosylation - Ethan Goddard-Borger
- Discovery and biosynthesis of ribosomally synthesized and posttranslationally modified peptides (RiPPs) - Qi Zhang
- Optical control of protein domain conformation and cell signaling - Harald Janovjak
- Chemoselective tyrosine bioconjugation of peptides and proteins through sulfate Click reaction - B. Moon Kim
- CXMS Analysis for Complex Protein Structures and Protein-Protein Interactions - Xiaoguang Lei
Tregear Award
5:15PM - 6:00PM
Wednesday, 11th September
Manhattan Room
Chair: Jackie Wilce
Dinner (Included)
6:00PM - 7:30PM
Wednesday, 11th September
Oak & Vine
Poster Session 2 and Drinks
7:30PM - 10:00PM
Wednesday, 11th September
Manhattan Room
Sponsored by:
- Synthesis and application of advanced fluorescent probes - Alejandra Gallardo-Godoy
- Detection of bioactive peptides including gonadotrophin-releasing factors (GnRHs) in horse urine using ultra-high performance liquid chromatography-high resolution mass spectrometry (UHPLC-HRMS) - Karen Y. Kwok
- Photooxidation of oxazoles – a new approach to solid-phase peptide synthesis - Chloe N. Larcombe
- Development of novel relaxin-3 analogues for blood-brain barrier penetration - Han Siean Lee
- Phosphorylation of α-synuclein induces distinct strains and propagation properties - Chuqiao Liang
- Dichloroacetone – A robust approach to acetone-linked bicyclic dimer peptides - Qingqing (Irene) Lin
- Synthesis of Peptide Natural Products Enabled by New Strategies for Late-Stage Modification - Yutong Lin
- The role of charge regulation in the interaction between oligo-peptides and polyelectrolytes - Raju Lunkad
- Insulin fatty acid acylation scan: Discovery of Insulin 327, an acylated hepato-preferential insulin analogue with high insulin receptor affinity - Peter Madsen
- Robust methodology for assembling peptides with tryptophan C-mannosylation - Runyu Mao
- Peptide modulating tension in cell membranes: the regulation of cell movement and morphology via actin remodeling - Toshihiro Masuda
- Tyrosine sulfation is an important post-translational modification in anti-inflammatory peptides from blood-feeding organisms. - Joshua W Maxwell
- The New Kid On The Block: Discovery and development of NaV channel inhibitor and µ-conotoxin NgIIIA - Kirsten L McMahon
- Peptide cyclisation using a pyridine-2,6-dicarbonitrile linker - Richard Morewood
- Structure-activity study of the analgesic NaV1.7 inhibiting venom peptide Pn3a - Alexander Mueller
- Chemical strategies to tune potency, selectivity and stability of neuropeptides - Markus Muttenthaler
- Design and synthesis of a PD-1 binding peptide and evaluation of its anti-tumor activity - Peiwei Yang
- A Zn(II)-catalyst permits bis-thioether peptide stapling under non-basic conditions - Huy Nguyen
- Noncanonical peptides as probes and inhibitors for flavivirus proteases - Christoph Nitsche
- Identification and Optimisation of a Lead Bromodomain Inhibitor - Alexander R Norman
- Membrane-bound structure and membrane selectivity of cationic antimicrobial peptide Hymenochirin-1Pa and its D9K analog - Akifumi Oyama
- Evaluation of biological activity of frog skin-derived peptide, ranatensin - Liliana Mrs. Palczynska
- Thiol-cyanobenzothiazole ligation: an efficient preparation of peptide-oligonucleotide conjugates - Nitin A Patil
- The Structural Features of an Ancient Peptide Family Buried within Vicilin Precursors. - Colton D. Payne
- Cyclic peptide conjugates: their mode-of action and interaction with cell membranes - Gregoire Philippe
- Cyclic peptides to probe the internal interactome of PDZ domains - Javier Rodriguez Balboa
- Decoding the complex regulation of cone snail venoms: connecting evolution and drug discovery - Himaya S.W.A.
- Novel methods for inhibiting amyloidogenesis in the presence of peptides in order to block hydrophobic interaction - Masatoshi Saiki
- Cytosolic Delivery of Macromolecules by Endosomolytic Cationic Helical Peptide - Kentarou Sakamoto
- Exploring the oxytocin receptor as a novel target for breast cancer - Cristina Sanchez de la Rosa
- Affinity-based functionalization of biomedical polymeric micelles through polymer-binding peptides - Toshiki Sawada
- Backbone cyclization of native α-conotoxin CIA: Influences on structure and bioactivity - Casey Schmidt
- The use of peptide-membrane interactions in the design of selective and potent sodium channel inhibitors - Christina Schroeder
- Discovery of tight binding inhibitors of hip1 a mycobacterium tuberculosis drug target - Nicholas C Schuman
- Conformational diversity in the neurotensin peptide upon binding neurotensin receptor 1 may drive receptor activation - Daniel J Scott
- Discovery and mechanistic investigations of ultrashort amphiphilic peptides that exhibit potent inhibition of Cryptococcus neoformans - Komal Sharma
- Tripeptide-induced mechanical property modulation of mesenchymal stem cells stimulates proliferation and wound healing - Swati Sharma
- Enhancing activity by combining antimicrobial peptides and antibiotics - Dean Sheard
- Evolving Peptide G Protein-Coupled Receptors (GPCRs) to Facilitate Structural Studies Using a Novel Lentiviral Based Method of Directed Evolution - Jonathan Siah
- Peptide based hydrogen sulfide responsive nanostructures for biomedical applications - Narendra Singh
- Analysis of granulin peptide folding - Rozita Takjoo
- Synthesis and biological activity of celogentin analogues - Varsha Thombare
- Iterative optimization of the cyclic peptide SFTI-1 yields potent inhibitors of neutrophil proteinase 3 - SIXIN ST TIAN
- Taking active steps to improving the pharmacokinetics of disulfide-rich peptides - Benjamin J Tombling
- μ‐Conotoxin KIIIA isomer selectivity on human voltage gated sodium channels - Hue N T Tran
- Enzymatic ligation of Nav1.7-inhibiting gating modifier and pore blocker toxins - Poanna Tran
- Exploration of amyloidogenic core β-sheet and the FEL-mediated dissociation of amyloid fibrils in SAA - Tomomi Ueda
- The characterization of triglyceride-based nanodroplets and their interaction with lipid specific peptides and proteins - Valerija Vezočnik
- A fluorescent protein-tagged peptide toxin as a tool for KV1.3 visualisation - Dorothy C. Wai
- Combinatorial peptide libraries in venoms of Australian nettle caterpillars - Andrew A Walker
- From sunflower to skin cancer: Development of melanocortin receptor-1 agonists based on the cyclic peptide framework of sunflower trypsin inhibitor-1 - Andrew M White
- Development of a lentiviral nanobody screening platform against peptide GPCRs - Lisa M Williams
- Delivery of a peptide-based vaccine against Group A Streptococcus with the help of cell penetrating peptides - Jieru Yang
- Anchoring epitopes to improve grafted peptide structure and activity - Huawu Yin
- A*STAR Peptide Engineering Platform (PEP): Targeting Macrocyclic Modalities for Protein-Protein Interactions - Tsz Ying Yuen
- In-cell structure determination of an antimicrobial peptide by DNP solid-state NMR - shiying zhu
- Peptidomimetics targeting the SOCS-SH2 domain - Hao Chen
- Receptor-Mediated MAPK and Akt Signaling are Maintained in Gamma-Irradiated FroZen Cells - Shima Hamidi
- Synthesis and Evaluation of a Library of Self-Adjuvanting Peptide and Protein Vaccines against Mycobacterium tuberculosis - Cameron Hanna
- Development of a single-chain peptide agonist for the G-protein-coupled receptor, RXFP1 - Praveen Praveen
- Improving in vivo analgesia through glycosylation of bilorphin, a biased μ-opioid derived from a novel tetrapeptide class found in an Australian fungus - Zoltan Dekan